Term Name: kenpaullone
Synonyms: 9-bromo-7,12-dihydroindolo[3,2-d][1]benzazepin-6(5H)-one, 9-bromopaullone
Definition: An indolobenzazepine that is paullone in which the hydrogen at position 9 is replaced by a bromo substituent. It is an ATP-competitive inhibitor of cyclin-dependent kinases (CDKs) and glycogen synthase kinase 3beta (GSK3beta).
Ontology: ChEBI [CHEBI:92658]  ( EBI )

Relationships
is a type of: indolobenzazepine lactam organobromine compound
has_functional_parent: paullone
has_role: cardioprotective agent EC 2.7.11.22 (cyclin-dependent kinase) inhibitor EC 2.7.11.26 (tau-protein kinase) inhibitor geroprotector